A simple solid phase diversity linker strategy using enol phosphonates

Campbell, I.B.; Guo, J.; Jones, E.; Steel, P.G.

doi:10.1039/b411111g

A simple solid phase diversity linker strategy using enol phosphonates

Campbell, I.B.; Guo, J.; Jones, E.; Steel, P.G.

Authors

I.B. Campbell

J. Guo

E. Jones

Professor Patrick Steel p.g.steel@durham.ac.uk
Professor

Abstract

Polymer bound lactam enol phosphonates can be easily generated using simple phenol on polystyrene resin. These stable, storable compounds can be released in a diversity cleavage strategy, using Suzuki cross coupling conditions, to provide 2-arylenamides in moderate to good overall yields.

Citation

Campbell, I., Guo, J., Jones, E., & Steel, P. (2004). A simple solid phase diversity linker strategy using enol phosphonates. Organic and Biomolecular Chemistry, 2(19), 2725-2727. https://doi.org/10.1039/b411111g

Journal Article Type	Article
Publication Date	2004-09
Deposit Date	Apr 19, 2007
Journal	Organic and Biomolecular Chemistry
Print ISSN	1477-0520
Electronic ISSN	1477-0539
Publisher	Royal Society of Chemistry
Peer Reviewed	Peer Reviewed
Volume	2
Issue	19
Pages	2725-2727
DOI	https://doi.org/10.1039/b411111g